Expert Opin Drug Saf 4(4):689706
However, the main concern with oral delivery is bioavailability, or how much of the peptide is absorbed into the bloodstream after digestion
10 mg Vial Reconstitution BAC water added 2 mL Concentration 5,000 mcg/mL 250 mcg dose volume 0.05 mL = 5 units 500 mcg dose volume 0.10 mL = 10 units Doses per vial at 250 mcg 40 BAC water added 3 mL Concentration 3,333 mcg/mL 250 mcg dose volume 0.075 mL = ~7.5 units 500 mcg dose volume 0.15 mL = 15 units Doses per vial at 250 mcg 40 Units shown are U-100 insulin syringe units (where 100 units = 1.0 mL)
As a defined small molecule, 5-Amino-1MQ is a "tool compound" in the classical pharmacology sense useful for probing NNMT biology specifically
Clean the injection site with alcohol, pinch the skin to create a fold of tissue, insert the needle at a 45-90 degree angle, inject slowly, and withdraw the needle
That last clause is the one that distinguishes a prescription peptide from a supplement